BMS794833 inhibits macrophage efferocytosis by directly binding to MERTK and inhibiting its activity.
Bae SH, Kim JH, Park TH, Lee K, Lee BI, Jang H
Exp Mol Med. 2022 Sep;54(9):1450-1460. doi: 10.1038/s12276-022-00840-x. Epub 2022 Sep 2.
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Plasmids from Article
| ID | Plasmid | Purpose |
|---|---|---|
| 196447 | pETDuet-MerTK_KRmutant-PTPN1 | Expression of MerTK Kinase Domain in E. coli and surface entropy reduction mutant for crystallization, coexpress PTPN1 |
| 197988 | pETDuet-MerTK-PTPN1 | Expression of MerTK Kinase Domain (wild-type) in E. coli |