GLP1R-Tango Citations (8)

Originally described in: PRESTO-Tango as an open-source resource for interrogation of the druggable human GPCRome.
Kroeze WK, Sassano MF, Huang XP, Lansu K, McCorvy JD, Giguere PM, Sciaky N, Roth BL Nat Struct Mol Biol. 2015 May;22(5):362-9. doi: 10.1038/nsmb.3014. Epub 2015 Apr 20. PubMed Journal

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Articles Citing GLP1R-Tango

Articles
Pancreatic alpha Cell-Derived Glucagon-Related Peptides Are Required for beta Cell Adaptation and Glucose Homeostasis. Traub S, Meier DT, Schulze F, Dror E, Nordmann TM, Goetz N, Koch N, Dalmas E, Stawiski M, Makshana V, Thorel F, Herrera PL, Boni-Schnetzler M, Donath MY. Cell Rep. 2017 Mar 28;18(13):3192-3203. doi: 10.1016/j.celrep.2017.03.005. PubMed
Agonist-induced membrane nanodomain clustering drives GLP-1 receptor responses in pancreatic beta cells. Buenaventura T, Bitsi S, Laughlin WE, Burgoyne T, Lyu Z, Oqua AI, Norman H, McGlone ER, Klymchenko AS, Correa IR Jr, Walker A, Inoue A, Hanyaloglu A, Grimes J, Koszegi Z, Calebiro D, Rutter GA, Bloom SR, Jones B, Tomas A. PLoS Biol. 2019 Aug 20;17(8):e3000097. doi: 10.1371/journal.pbio.3000097. eCollection 2019 Aug. PubMed
Dimerization/oligomerization of the extracellular domain of the GLP-1 receptor and the negative cooperativity in its ligand binding revealed by the improved NanoBiT. Song X, Yu Y, Shen C, Wang Y, Wang N. FASEB J. 2020 Mar;34(3):4348-4368. doi: 10.1096/fj.201902007R. Epub 2020 Jan 23. PubMed
The Influence of Peptide Context on Signaling and Trafficking of Glucagon-like Peptide-1 Receptor Biased Agonists. Fang Z, Chen S, Pickford P, Broichhagen J, Hodson DJ, Correa IR Jr, Kumar S, Gorlitz F, Dunsby C, French PMW, Rutter GA, Tan T, Bloom SR, Tomas A, Jones B. ACS Pharmacol Transl Sci. 2020 Mar 17;3(2):345-360. doi: 10.1021/acsptsci.0c00022. eCollection 2020 Apr 10. PubMed
Recombinant Peptide Production Platform Coupled with Site-Specific Albumin Conjugation Enables a Convenient Production of Long-Acting Therapeutic Peptide. Bak M, Park J, Min K, Cho J, Seong J, Hahn YS, Tae G, Kwon I. Pharmaceutics. 2020 Apr 16;12(4). pii: pharmaceutics12040364. doi: 10.3390/pharmaceutics12040364. PubMed
Signalling, trafficking and glucoregulatory properties of glucagon-like peptide-1 receptor agonists exendin-4 and lixisenatide. Pickford P, Lucey M, Fang Z, Bitsi S, de la Serna JB, Broichhagen J, Hodson DJ, Minnion J, Rutter GA, Bloom SR, Tomas A, Jones B. Br J Pharmacol. 2020 Sep;177(17):3905-3923. doi: 10.1111/bph.15134. Epub 2020 Jun 19. PubMed
GRK2 regulates GLP-1R-mediated early phase insulin secretion in vivo. Arcones AC, Vila-Bedmar R, Mirasierra M, Cruces-Sande M, Vallejo M, Jones B, Tomas A, Mayor F Jr, Murga C. BMC Biol. 2021 Mar 3;19(1):40. doi: 10.1186/s12915-021-00966-w. PubMed
Effect of C-terminus Conjugation via Different Conjugation Chemistries on In Vivo Activity of Albumin-Conjugated Recombinant GLP-1. Park J, Bak M, Min K, Kim HW, Cho JH, Tae G, Kwon I. Pharmaceutics. 2021 Feb 15;13(2). pii: pharmaceutics13020263. doi: 10.3390/pharmaceutics13020263. PubMed

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